Melatonin suppresses the induction of AP-1 transcription factor components in the pars tuberalis of the pituitary

Mol Cell Endocrinol. 1996 Oct 14;123(1):71-80. doi: 10.1016/0303-7207(96)03897-x.

Abstract

In ovine pars tuberalis cells which express high affinity Mel 1a melatonin receptors, the ability of melatonin to directly stimulate or inhibit AP-1 transcription factor gene expression was studied. Effects of melatonin upon mRNA expression by forskolin, serum and IGF-1 were also investigated. Northern analysis showed melatonin had no direct stimulatory nor inhibitory effect upon transcription or translation. Melatonin was able to significantly inhibit forskolin-stimulated induction of c-fos and jun B mRNA whilst forskolin had no effect upon c-jun or jun D. Induction of c-Fos translation by forskolin was also inhibited by melatonin. Serum induced c-fos and c-jun, but melatonin was unable to affect these changes. Similarly IGF-1 stimulated c-fos and melatonin had no effect upon this induction. From these results it can be concluded that melatonin has no independent effects on expression of the AP-1 genes, rather its primary function is to inhibit cell activities through cyclic AMP-dependent routes of gene activation.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Animals
  • Base Sequence
  • Blotting, Northern
  • Cells, Cultured
  • Colforsin / pharmacology
  • Female
  • Gene Expression / drug effects
  • Genes, jun / drug effects
  • In Situ Hybridization
  • Insulin-Like Growth Factor I / pharmacology
  • Male
  • Melatonin / pharmacology*
  • Oligonucleotide Probes
  • Pituitary Gland, Anterior / cytology
  • Pituitary Gland, Anterior / drug effects
  • Pituitary Gland, Anterior / metabolism*
  • Proto-Oncogene Proteins c-jun / biosynthesis
  • RNA, Messenger / biosynthesis
  • Sheep
  • Transcription Factor AP-1 / biosynthesis*
  • Transcription, Genetic / drug effects*

Substances

  • Oligonucleotide Probes
  • Proto-Oncogene Proteins c-jun
  • RNA, Messenger
  • Transcription Factor AP-1
  • Colforsin
  • Insulin-Like Growth Factor I
  • Melatonin