PC-2, linear homoglucan with alpha-linkages, peripherally enhances the hippocampal long-term potentiation

Pharm Res. 1996 Sep;13(9):1322-6. doi: 10.1023/a:1016009630329.

Abstract

Purpose: To investigate central effectiveness of PC-2, a glucan from lichen Parmelia caperata with alpha(1-3)(1-4) linkages in the ratio 3:2, with regard to the long-term potentiation (LTP) of evoked potential.

Methods: The extent of LTP, induced by high-frequency stimulation of medial perforant pathway, was evaluated as fractional increase in population spike amplitude in dentate gyrus in anesthetized rats.

Results: Oral and intravenous application of PC-2 resulted in significant enhancement of LTP elicited by a weak, but not by a strong, tetanic stimulation. No influence of PC-2 on basal evoked synaptic potential was found. Bilateral adrenalectomy profoundly suppressed the positive impact of the glucan on the formation of LTP, but showed no effect upon the magnitude and time-course of population spike enhancement in vehicle-treated subjects. Two related alpha-glucans with different chemical structures did not show any effect comparable to that of PC-2.

Conclusions: Peripheral application of PC-2 significantly enhances LTP in dentate gyrus in rats. Results indicate that the effect of PC-2 might be peripherally mediated and that the specific higher structure of PC-2 is crucial for its biological activity.

MeSH terms

  • Adrenalectomy
  • Animals
  • Carbohydrate Sequence
  • Dentate Gyrus / drug effects*
  • Dentate Gyrus / physiology
  • Evoked Potentials
  • Glucans / isolation & purification
  • Glucans / pharmacology*
  • Lichens / chemistry
  • Long-Term Potentiation / drug effects*
  • Male
  • Molecular Sequence Data
  • Polysaccharides / administration & dosage
  • Polysaccharides / isolation & purification
  • Polysaccharides / pharmacology*
  • Rats
  • Rats, Wistar

Substances

  • Glucans
  • Polysaccharides
  • glucan PC-2