Fast desensitizing kainate-gated current resolved in whole-cell experiments on isolated rat hippocampal neurons

Eur J Pharmacol. 1996 May 6;303(1-2):145-9. doi: 10.1016/0014-2999(96)00143-4.

Abstract

In whole-cell concentration-jump experiments on dissociated rat hippocampal neurons the existence of a fast desensitizing component of a kainate-gated current was demonstrated. More than 90% of all neurons tested possessed such a receptor. Electrophysiological and pharmacological data suggest an association of this fast kainate-gated current with that mediated through a combination of subunits forming a low-affinity "(RS)-alpha-amino-3-hydroxy-5-methyl-4-isoxazolopropionic acid (AMPA)-preferring' receptor. Kinetic data suggest the existence of a compact spatial location of fast desensitizing "AMPA-preferring' receptors which are naturally expressed on the surface of the neurons. An AMPA-insensitive current component mediated through fast desensitizing high-affinity kainate receptors was not observed.

Publication types

  • Comparative Study

MeSH terms

  • Animals
  • Benzothiadiazines / pharmacology
  • Cells, Cultured
  • Concanavalin A / pharmacology
  • Dose-Response Relationship, Drug
  • Excitatory Amino Acid Agonists / pharmacology*
  • Hippocampus / drug effects*
  • Hippocampus / physiology*
  • Kainic Acid / pharmacology*
  • Male
  • Patch-Clamp Techniques
  • Rats

Substances

  • Benzothiadiazines
  • Excitatory Amino Acid Agonists
  • Concanavalin A
  • cyclothiazide
  • Kainic Acid