Abstract
Micromolar concentrations of hydrogen peroxide induced the phosphorylation of mitogen-activated protein (MAP) kinases and a lethal response in growth-arrested smooth muscle cells (A7r5). The H202-induced phosphorylation of MAP-kinases was markedly lower in the presence of protein tyrosine kinase (PTK) inhibitors or in protein kinase C (PKC) down-regulated cells. Similarly, the toxicity of H202 was diminished by concomitant addition of either PKC or PTK inhibitors and was also lower in PKC down-regulated cells. These results are consistent with the possibility that phosphorylation of MAP-kinases is a critical event in the toxic response of cultured smooth muscle cells to H202.
Publication types
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Research Support, Non-U.S. Gov't
MeSH terms
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Animals
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Calcium-Calmodulin-Dependent Protein Kinases / metabolism*
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Catechols / pharmacology
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Cell Death / drug effects
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Cell Division / drug effects
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Clone Cells
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Down-Regulation
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Electrophoresis, Polyacrylamide Gel
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Enzyme Inhibitors / pharmacology
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Hydrogen Peroxide / pharmacology*
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Muscle, Smooth / cytology*
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Muscle, Smooth / drug effects
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Naphthalenes / pharmacology
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Nitriles / pharmacology
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Phosphorylation
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Protein Kinase C / antagonists & inhibitors
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Protein Kinase C / metabolism
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Protein-Tyrosine Kinases / antagonists & inhibitors
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Rats
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Tyrphostins*
Substances
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Catechols
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Enzyme Inhibitors
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Naphthalenes
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Nitriles
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Tyrphostins
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calphostin complex
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Hydrogen Peroxide
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Protein-Tyrosine Kinases
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Protein Kinase C
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Calcium-Calmodulin-Dependent Protein Kinases
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tyrphostin A23