Crystallographic evidence that the F2 kringle catalytic domain linker of prothrombin does not cover the fibrinogen recognition exosite

J Biol Chem. 1996 Feb 16;271(7):3413-6. doi: 10.1074/jbc.271.7.3413.

Abstract

The 2.6-A x-ray crystal structure of bovine alpha-thrombin in complex with rhodniin, a protein inhibitor isolated from the bug Rhodnius prolixus, has been solved and refined. The structure has enabled us to trace the N-terminal part of the 49-residue A-chain of bovine alpha-thrombin for the first time, which is fixed in a U-shaped loop on the molecular surface opposite the active site canyon. Model building shows that the 25 amino acid residues that link the A-chain and F2 kringle cannot run through the fibrinogen recognition exosite. This demonstrates that this fibrinogen recognition exosite is available in prothrombin and meizothrombin.

Publication types

  • Comparative Study

MeSH terms

  • Amino Acid Sequence
  • Animals
  • Binding Sites
  • Cattle
  • Crystallography, X-Ray
  • Fibrinogen / metabolism*
  • Humans
  • Insect Hormones / metabolism
  • Insect Proteins*
  • Kringles*
  • Models, Molecular
  • Molecular Sequence Data
  • Protein Structure, Secondary*
  • Prothrombin / chemistry*
  • Prothrombin / metabolism*
  • Sequence Homology, Amino Acid
  • Serine Proteinase Inhibitors / metabolism
  • Vertebrates

Substances

  • Insect Hormones
  • Insect Proteins
  • Serine Proteinase Inhibitors
  • rhodniin protein, Rhodnius
  • Prothrombin
  • Fibrinogen