Neuroprotective effects of NBQX on hypoxia-induced neuronal damage in rat hippocampus

Neuroreport. 1995 Nov 13;6(16):2205-8. doi: 10.1097/00001756-199511000-00025.

Abstract

Models of cerebral ischaemia were used for analysis of mechanism of neuronal cell death and/or damage. Ischaemia is caused dominantly by severe hypoxia and hypoglycaemia: in the present study, we examined the influence of severe in vivo hypoxia (5% O2/95% N2 for 30 min at 22 degrees C). After hypoxia, neuronal damage was observed in the CA3 and dentate gyrus (DG) after 3 and 21 days of survival, but not in the CA1.2,3-Dihydroxy-6-nitro-7-sulphamoyl-benzo(F)quinoxaline (NBQX), an antagonist for AMPA/kainate receptors, showed neuroprotective effects in the CA3 and DG. These results suggest that hypoxia may induce neuronal damage in the CA3 and DG through activation of AMPA/kainate receptors.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Analysis of Variance
  • Animals
  • Excitatory Amino Acid Antagonists / pharmacology*
  • Hippocampus / drug effects*
  • Hippocampus / pathology
  • Histocytochemistry
  • Hypoxia, Brain / pathology
  • Male
  • Neurons / drug effects
  • Neuroprotective Agents / pharmacology*
  • Quinoxalines / pharmacology*
  • Rats
  • Rats, Inbred F344
  • Receptors, AMPA / antagonists & inhibitors*
  • Receptors, Kainic Acid / antagonists & inhibitors*

Substances

  • Excitatory Amino Acid Antagonists
  • Neuroprotective Agents
  • Quinoxalines
  • Receptors, AMPA
  • Receptors, Kainic Acid
  • 2,3-dioxo-6-nitro-7-sulfamoylbenzo(f)quinoxaline