Evidence for competition between vitamin K-dependent clotting factors for intracellular processing by the vitamin K-dependent gamma-carboxylase

Thromb Res. 1995 Oct 1;80(1):63-73. doi: 10.1016/0049-3848(95)00151-g.

Abstract

This study demonstrates an apparent competition between newly synthesized precursors of prothrombin and factor X for binding to and processing by the gamma-carboxylase in the ER membrane of hepatocytes. The precursor of factor X appears to exhibit a strong affinity for the carboxylase than the prothrombin precursor. This conclusion is supported by the findings that 1) in normal hepatocytes, the factor X precursor prevents increased prothrombin precursor binding to the ER membrane, 2) increased prothrombin binding to the ER membrane was measured in H4-II-E-C3 Reuber H-35 cells where factor X synthesis is suppressed. The variations in the concentrations of the prothrombin and the factor X precursors that were as associated with the ER membrane correlated with the available prothrombin and factor X substrate pools for the gamma-carboxylase.

Publication types

  • Research Support, U.S. Gov't, P.H.S.

MeSH terms

  • Animals
  • Anticoagulants / pharmacology
  • Base Sequence
  • Blotting, Western
  • Carboxy-Lyases / metabolism*
  • Endoplasmic Reticulum / drug effects
  • Endoplasmic Reticulum / metabolism*
  • Factor X / biosynthesis*
  • Factor X / drug effects
  • Liver Neoplasms, Experimental
  • Molecular Sequence Data
  • Prothrombin / biosynthesis*
  • Prothrombin / drug effects
  • RNA, Messenger / analysis
  • Rats
  • Tumor Cells, Cultured
  • Vitamin K / metabolism*
  • Warfarin / pharmacology

Substances

  • Anticoagulants
  • RNA, Messenger
  • Vitamin K
  • Warfarin
  • Prothrombin
  • Factor X
  • Carboxy-Lyases

Associated data

  • GENBANK/X79807