Protective effect of clonazepam on ischemic brain damage induced by 10-minute bilateral carotid occlusion in Mongolian gerbils

Funct Neurol. 1993 Mar-Apr;8(2):115-20.

Abstract

A 10-min bilateral carotid occlusion (BCO) in a control group of Mongolian gerbils, induced a transient generalized epileptic activity both in the hippocampal and in the cortical regions, associated with motor manifestations. After recirculation, spiking activity persisted, reaching its maximum peak within 18-36 h and then slowly decreasing till its total disappearance on the 6th-7th day. On the 7th day, histological studies manifested a selective loss of CA1 hippocampal neurons. The treated gerbils (divided in 2 groups according to the dosage used) were administered clonazepam (CZP), a benzodiazepine receptor agonist, immediately after clamping and again every 24 h for the following three days at dosages of 0.05 and 0.1 mg/kg i.p., respectively. The drug inhibited epileptic activity in a dose-dependent manner, while it prevented CA1 neuronal loss at both doses. These results point to a possible derangement of the GABAergic system which probably in turn triggers an exaggerated excitation.

MeSH terms

  • Animals
  • Brain Ischemia / metabolism*
  • Brain Ischemia / physiopathology
  • Carotid Arteries / drug effects
  • Carotid Arteries / physiopathology*
  • Clonazepam / pharmacology*
  • Epilepsy / metabolism
  • Epilepsy / physiopathology
  • Gerbillinae*
  • Hippocampus / drug effects
  • Hippocampus / physiopathology
  • Hippocampus / ultrastructure
  • Nerve Degeneration

Substances

  • Clonazepam