Pharmacological aspects of R-(+)-7-OH-DPAT, a putative dopamine D3 receptor ligand

Eur J Pharmacol. 1993 Nov 16;249(3):R9-10. doi: 10.1016/0014-2999(93)90533-n.

Abstract

The R-(+)-isomer of 7-hydroxy-2-(N,N-di-n-propylamino)tetralin (7-OH-DPAT) bound with a more than 200-fold higher affinity to cloned human dopamine D3 receptors (Ki = 0.57 nM) than to dopamine D2 receptors; the corresponding S-(-)-enantiomer had considerably less affinity for both dopamine receptor subtypes, indicating that the known enantiomer selectivity of 7-OH-DPAT for the 'classical' dopamine D2 receptor subtype extends to the recently discovered dopamine D3 receptor subtype. In rats R-(+)-7-OH-DPAT dose dependently (10-1000 nmol/kg) decreased dopamine release and induced yawning, while sniffing behaviour occurred at the highest dose tested (1000 nmol/kg). The possibility that the inhibition of dopamine release and the elicitation of yawning are mediated by dopamine D3 receptors is considered.

MeSH terms

  • Animals
  • Behavior, Animal / drug effects*
  • Dopamine / metabolism
  • Dose-Response Relationship, Drug
  • Male
  • Rats
  • Rats, Wistar
  • Receptors, Dopamine / drug effects
  • Receptors, Dopamine / metabolism*
  • Receptors, Dopamine D2*
  • Receptors, Dopamine D3
  • Stereoisomerism
  • Tetrahydronaphthalenes / metabolism
  • Tetrahydronaphthalenes / pharmacology*
  • Yawning / drug effects

Substances

  • Drd3 protein, rat
  • Receptors, Dopamine
  • Receptors, Dopamine D2
  • Receptors, Dopamine D3
  • Tetrahydronaphthalenes
  • 7-hydroxy-2-N,N-dipropylaminotetralin
  • Dopamine