Dideoxynucleoside resistance emerges with prolonged zidovudine monotherapy. The RV43 Study Group

Antimicrob Agents Chemother. 1994 Feb;38(2):307-14. doi: 10.1128/AAC.38.2.307.

Abstract

Human immunodeficiency virus type 1 (HIV-1) isolates resistant to zidovudine (ZDV) have previously been demonstrated to exhibit in vitro cross-resistance to other similar dideoxynucleoside agents which contain a 3'-azido group. However, cross-resistance to didanosine (ddI) or dideoxycytidine (ddC) has been less well documented. ZDV, ddI, and ddC susceptibility data have been collected from clinical HIV-1 isolates obtained by five clinical centers and their respective retrovirology laboratories. All subjects were treated only with ZDV. Clinical HIV-1 isolates were isolated, amplified, and assayed for drug susceptibility in standardized cultures of phytohemagglutinin-stimulated donor peripheral blood mononuclear cells obtained from healthy seronegative donors. All five cohorts showed a correlation between decreased in vitro susceptibility to ZDV and decreased susceptibility to ddI and ddC. For each 10-fold decrease in ZDV susceptibility, an average corresponding decrease of 2.2-fold in ddI susceptibility was observed (129 isolates studied; P < 0.001, Fisher's test of combined significance). Similarly, susceptibility to ddC decreased 2.0-fold for each 10-fold decrease in ZDV susceptibility (82 isolates studied; P < 0.001, Fisher's test of combined significance). These data indicate that a correlation exists between HIV-1 susceptibilities to ZDV and ddI or ddC for clinical HIV-1 isolates.

Publication types

  • Research Support, Non-U.S. Gov't
  • Research Support, U.S. Gov't, Non-P.H.S.
  • Research Support, U.S. Gov't, P.H.S.

MeSH terms

  • AIDS-Related Complex / blood
  • Acquired Immunodeficiency Syndrome / blood
  • Didanosine / pharmacology*
  • Drug Resistance, Microbial
  • HIV Seropositivity / blood
  • HIV-1 / drug effects*
  • Humans
  • Leukocytes, Mononuclear / microbiology
  • Microbial Sensitivity Tests
  • Time Factors
  • Zalcitabine / pharmacology*
  • Zidovudine / pharmacology*

Substances

  • Zidovudine
  • Zalcitabine
  • Didanosine