Mechanism of prolactin action on the dissociation of prolactin from rabbit mammary gland receptor

Biochem Biophys Res Commun. 1994 Aug 15;202(3):1395-9. doi: 10.1006/bbrc.1994.2085.

Abstract

In order to elucidate the action of prolactin (PRL) on the dissociation of PRL from the receptor, Triton-solubilized and concanavalin A-purified rabbit mammary gland PRL receptor was immobilized onto a nitrocellulose membrane, and the dissociation of PRL was determined in the presence of PRL. PRL accelerated the dissociation of PRL in a concentration dependent manner for the first 3 h of incubation. The effects of PRL on dissociation were independent of the occupancy of PRL at the zero-time dissociation. In particular, PRL-dependency was influenced by the PRL-binding capacity of the membrane. The dissociation reaction was PRL-independent in the low-binding capacity membrane, indicating that PRL itself had no accelerating actions. With greater binding capacity, the dissociation reaction was seen to become PRL-dependent. It was concluded that PRL accelerated the dissociation of PRL through the formation of PRL-receptor complex when the receptor was located closely to the neighboring receptors.

MeSH terms

  • Animals
  • Binding Sites
  • Female
  • Growth Hormone / physiology
  • Luteinizing Hormone / physiology
  • Mammary Glands, Animal / metabolism*
  • Prolactin / physiology*
  • Rabbits
  • Receptors, Prolactin / metabolism*
  • Thyrotropin / physiology

Substances

  • Receptors, Prolactin
  • Prolactin
  • Luteinizing Hormone
  • Thyrotropin
  • Growth Hormone