[Antifertility effects of mifepristone and epostane alone and in combination in rats]

Zhongguo Yao Li Xue Bao. 1993 Sep;14(5):437-40.
[Article in Chinese]

Abstract

A complete interceptive action on pregnancy was shown after ig mifepristone (RU-486) 16 mg.kg-1 or epostane 96 mg.kg-1 on d 10 of pregnancy in rats. The ig ED50 (95% fiducial limits) of RU-486 when given alone and in combination with epostane 12 mg.kg-1 were found to be 7.8 (5.3-10.0) and 2.6 (2.0-3.3) mg.kg-1, respectively (P < 0.05), while those of epostane when given alone and in combination with RU-486 4 mg.kg-1 were 25.5 (19.4-33.6) and 5.6 (4.7-7.4) mg.kg-1, respectively (P < 0.05). An absorption promotor, sodium dodecyl sulfate 24 mg.kg-1 ig, when given in combination with RU-486 8 mg.kg-1 or epostane 24 mg.kg-1, induced complete interceptive action on pregnancy. Levels of plasma progesterone declined significantly when epostane 12 mg.kg-1 was given in combination with RU-486 4 mg.kg-1 as compared with epostane 12 mg.kg-1 alone (P < 0.05). Results showed that drug combination therapy was of benefit both to RU-486 and epostane in their interceptive actions.

Publication types

  • English Abstract

MeSH terms

  • Abortifacient Agents, Steroidal / pharmacology*
  • Abortion, Induced
  • Androstenols / pharmacology*
  • Animals
  • Drug Synergism
  • Female
  • Fertility / drug effects*
  • Mice
  • Mice, Inbred ICR
  • Mifepristone / pharmacology*
  • Pregnancy
  • Random Allocation
  • Rats
  • Rats, Sprague-Dawley
  • Sodium Dodecyl Sulfate / pharmacology

Substances

  • Abortifacient Agents, Steroidal
  • Androstenols
  • Mifepristone
  • Sodium Dodecyl Sulfate
  • epostane