Depletion of intracellular Ca2+ stores activates a maitotoxin-sensitive nonselective cationic current in beta-cells

J Biol Chem. 1994 Dec 23;269(51):32055-8.

Abstract

Glucose stimulation of beta-cell insulin secretion is initiated by membrane depolarization coupled with an elevation in intracellular Ca2+ concentration ([Ca2+]i). Both depolarization-dependent Ca2+ entry and intracellular Ca2+ store release contribute to the sugar-induced rise in [Ca2+]i. Here we show that maneuvers depleting intracellular Ca2+ stores induce membrane depolarization and a sustained nitrendipine-sensitive Ca2+ influx, whereas interventions promoting Ca2+ store refilling produce a hyperpolarization and inhibit Ca2+ influx. Both intracellular Ca2+ store depletion and maitotoxin activated a depolarizing nonselective cation current carried principally by Na+ in the physiological range of membrane potentials. The activation of such a current may form the paradigm by which excitable cells refill depleted intracellular Ca2+ stores by depolarization-driven opening of voltage-activated Ca2+ channels.

MeSH terms

  • Animals
  • Calcium / metabolism*
  • Calcium Channels / drug effects*
  • Calcium Channels / physiology
  • In Vitro Techniques
  • Islets of Langerhans / drug effects*
  • Islets of Langerhans / physiology
  • Marine Toxins / pharmacology*
  • Membrane Potentials
  • Mice
  • Mice, Inbred C57BL
  • Oxocins*

Substances

  • Calcium Channels
  • Marine Toxins
  • Oxocins
  • maitotoxin
  • Calcium