The conserved membrane-proximal region of an integrin cytoplasmic domain specifies ligand binding affinity

J Biol Chem. 1995 May 26;270(21):12411-7. doi: 10.1074/jbc.270.21.12411.

Abstract

Integrin affinities for ligands can change markedly via a process termed inside-out signaling. We expressed several truncations of the beta 3 cytoplasmic domain in conjunction with an "activating" alpha subunit chimera, alpha IIb alpha 6B. Deletion of the 4 C-terminal residues of the beta 2 tail blocked inside-out signaling as assessed by the binding of an activation-specific antibody, PAC1. Several additional truncations remained in the low affinity state, but complete truncation (beta 3 delta 717) caused PAC1 binding. Activation by this truncation mutant did not depend on the alpha subunit cytoplasmic domain and was resistant to inhibitors of cellular metabolism and the over-expression of an isolated beta 3 cytoplasmic domain. Since deletion of beta 3(Leu717-Asp723) results in a constitutively activated integrin, this membrane-proximal seven amino acids of the beta 3 cytoplasmic domain is required to maintain alpha IIb beta 3 in a default low affinity state. The amino acid sequence of this region is conserved among integrins. Moreover, the conserved membrane-proximal sequence in alpha subunit tails seems to serve a similar function. Consequently, the conserved membrane-proximal regions of both integrin cytoplasmic domains control the ligand binding affinity of the extracellular domain.

Publication types

  • Comparative Study
  • Research Support, Non-U.S. Gov't
  • Research Support, U.S. Gov't, P.H.S.

MeSH terms

  • Amino Acid Sequence
  • Animals
  • Antigens, CD / genetics
  • Antigens, CD / metabolism*
  • CHO Cells
  • Cell Polarity
  • Conserved Sequence
  • Cricetinae
  • DNA Mutational Analysis
  • Integrin beta3
  • Integrins / genetics
  • Integrins / metabolism*
  • Ligands
  • Molecular Sequence Data
  • Protein Binding
  • Protein Conformation
  • Recombinant Fusion Proteins / metabolism
  • Recombinant Proteins / metabolism
  • Sequence Deletion
  • Signal Transduction

Substances

  • Antigens, CD
  • Integrin beta3
  • Integrins
  • Ligands
  • Recombinant Fusion Proteins
  • Recombinant Proteins