Absorption behavior of sulpiride described using Weibull functions

Int J Clin Pharmacol Ther. 1995 May;33(5):299-303.

Abstract

Deconvolution absorption profiles of oral sulpiride formulations were calculated from plasma concentration-time data obtained in an open, 3-period study with a crossover of the 2 oral formulations in 12 healthy volunteers following single intravenous (100 mg) and oral (2 x 50 mg capsules, 200 mg tablets) application of sulpiride. A model based on 2 Weibull-functions, and applied using NONMEM, described the complex absorption profiles more satisfactorily than a first order absorption model or a model based on a single Weibull-function.

Publication types

  • Clinical Trial
  • Randomized Controlled Trial

MeSH terms

  • Absorption
  • Administration, Oral
  • Adult
  • Biological Availability
  • Capsules
  • Chromatography, High Pressure Liquid
  • Computer Simulation
  • Cross-Over Studies
  • Female
  • Humans
  • Injections, Intravenous
  • Male
  • Models, Chemical
  • Reference Standards
  • Sulpiride / administration & dosage
  • Sulpiride / blood
  • Sulpiride / pharmacokinetics*
  • Tablets

Substances

  • Capsules
  • Tablets
  • Sulpiride