[NONMEM approach for estimating population pharmacokinetic parameters of phenytoin in Chinese epileptics]

Yao Xue Xue Bao. 1995;30(3):172-8.
[Article in Chinese]

Abstract

Routine clinical pharmacokinetic data collected from epileptic out-patients who received phenytoin (PHT) were analysed to estimate population pharmacokinetic parameters. There were 258 steady-state serum phenytoin concentrations and associated dosage (mg.d-1) from 161 out-patients. The data were analysed using NONMEM program. The influence of body weight, drug combinations and sex on the maximum elimination rate (Vm) and age on the Michaelis-Menten constant (Km) were investigated. The Vm and Km of phenytoin in a 60 kg adult out-patient, without combination with other drugs (phenobarbital, clonazepam or diazepam) were estimated to be 439 mg.d-1 and 6.21 micrograms.ml-1, respectively. The best function adjusts Vm to the 0.57 power in proportion to body weight. The Km for patients less than 15 years old was 7% less than that for adults. The Vm of patients treated with phenytoin combined with phenobarbital, clonazepam or diazepam will increase 8.4 mg.d-1.

Publication types

  • English Abstract
  • Research Support, Non-U.S. Gov't

MeSH terms

  • Adolescent
  • Adult
  • Aged
  • Child
  • Child, Preschool
  • Epilepsy / metabolism*
  • Female
  • Humans
  • Male
  • Middle Aged
  • Models, Statistical
  • Phenytoin / pharmacokinetics*

Substances

  • Phenytoin