Phosphatidylethanolamine induces high affinity binding sites for factor VIII on membranes containing phosphatidyl-L-serine

J Biol Chem. 1995 Aug 4;270(31):18500-5. doi: 10.1074/jbc.270.31.18500.

Abstract

Synthetic membranes of phosphatidylcholine require inclusion of at least 5% phosphatidylserine (Ptd-L-Ser) to form binding sites for factor VIII. The relatively high requirement for Ptd-L-Ser suggests that stimulated platelets may contain another membrane constituent that enhances expression of factor VIII-binding sites. We report that phosphatidylethanolamine (PE), which is exposed in concert with Ptd-L-Ser in the course of platelet stimulation, induces high affinity binding sites for factor VIII on synthetic membranes containing 1-15% Ptd-L-Ser. The affinity of factor VIII for binding sites on membranes of Ptd-L-Ser/PE/phosphatidylcholine in a 4:20:76 ratio was 10.2 +/- 3.5 nM with 180 +/- 33 phospholipid molecules/site. PE did not induce binding sites on membranes of 4% Ptd-D-Ser, indicating that the induced binding sites require the correct stereochemistry of Ptd-L-Ser as well as PE. Egg PE and dimyristoyl-PE were equivalent for inducing factor VIII-binding sites, indicating that hexagonal phase-inducing properties of PE are not important. We conclude that PE induces high affinity factor VIII-binding sites on membranes with physiologic mole fractions of Ptd-L-Ser, possibly including those of stimulated platelets.

Publication types

  • Research Support, U.S. Gov't, Non-P.H.S.

MeSH terms

  • Binding Sites
  • Blood Platelets / metabolism
  • Factor VIII / metabolism*
  • Flow Cytometry
  • Fluorescent Dyes
  • Humans
  • Membranes, Artificial*
  • Phosphatidylethanolamines*
  • Phosphatidylserines* / chemistry
  • Recombinant Proteins / metabolism
  • Stereoisomerism
  • Structure-Activity Relationship

Substances

  • Fluorescent Dyes
  • Membranes, Artificial
  • Phosphatidylethanolamines
  • Phosphatidylserines
  • Recombinant Proteins
  • Factor VIII