Effect of three bile acid binding polymers on the biosynthesis of 14C-cholesterol from 14C-sodium acetate in the rat

Res Commun Chem Pathol Pharmacol. 1981 Aug;33(2):373-6.

Abstract

The relative activity of three bile acid binding polymers in increasing cholesterol biosynthesis in the rat from 14C-acetate was determined by measuring blood levels of 14C-cholesterol after intraperitoneally administered 14C-acetate. CAT-FLOC and 3,3-ionene were 4-5 times more active than cholestyramine in this study which correlated well with the results of hypocholesteremic testing in dogs.

MeSH terms

  • Acetates / metabolism*
  • Animals
  • Bile Acids and Salts / metabolism*
  • Cholesterol / biosynthesis*
  • Cholestyramine Resin / pharmacology
  • Polyethylenes*
  • Polymers / pharmacology
  • Quaternary Ammonium Compounds / pharmacology
  • Rats

Substances

  • Acetates
  • Bile Acids and Salts
  • Polyethylenes
  • Polymers
  • Quaternary Ammonium Compounds
  • Cholestyramine Resin
  • poly-N,N-dimethyl-N,N-diallylammonium chloride
  • 3,3-ionene
  • Cholesterol