Pyrrolnitrin analogues. VIII - Synthesis and antibacterial activity of new 1,4- and 1,5-diarylpyrroles

Farmaco Sci. 1983 Sep;38(9):630-9.

Abstract

From ethyl 1-aryl-2-methyl-4-(4-nitrophenyl)pyrrole-3-carboxylates new 1-aryl-2-methyl-4-(4-nitrophenyl)pyrrolderivatives wer prepared. These compounds and some previously reported 1,4- and 1,5-diarylpyrroles were subjected to in vitro antimicrobial screenings. Namely some 1-aryl-2-methyl-4-(4-nitrophenyl)pyrrole-3-carboxylic acids and its 5-chloroderivatives are the most potent. The results obtained are discussed on the basis of structure-activity relationships.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Anti-Bacterial Agents / chemical synthesis*
  • Bacteria / drug effects
  • Chemical Phenomena
  • Chemistry
  • Microbial Sensitivity Tests
  • Pyrroles / chemical synthesis*
  • Pyrroles / pharmacology

Substances

  • Anti-Bacterial Agents
  • Pyrroles