Quantitative structure-activity relationship in 1-substituted ureidophenoxy-3-amino-2-propanols, a class of beta-adrenergic blocking agents

Arzneimittelforschung. 1980;30(10):1613-7.

Abstract

The beta-adrenergic blocking potency of 56 1-substituted ureidophenoxy-3-amino-2-propanols has been analysed in terms of the linear Free-Wilson model. The values obtained for the Free-Wilson coefficients have been correlated with the chemico-physical parameters of the substituents. The preliminary indication given by the Free-Wilson analysis has been confirmed by a quantitative regression analysis, carried out in the frame of the "mixed approach" method.

MeSH terms

  • Adrenergic beta-Antagonists / pharmacology*
  • Chemical Phenomena
  • Chemistry, Physical
  • Propanolamines / pharmacology*
  • Regression Analysis
  • Structure-Activity Relationship

Substances

  • Adrenergic beta-Antagonists
  • Propanolamines