Therapeutic Potential of Oligo-Fucoidan in Mitigating Peritoneal Dialysis-Associated Fibrosis

Mar Drugs. 2024 Nov 25;22(12):529. doi: 10.3390/md22120529.

Abstract

Peritoneal dialysis (PD) serves as a home-based kidney replacement therapy with increasing utilization across the globe. However, long-term use of high-glucose-based PD solution incites repeated peritoneal injury and inevitable peritoneal fibrosis, thus compromising treatment efficacy and resulting in ultrafiltration failure eventually. In the present study, we utilized human mesothelial MeT-5A cells for the in vitro experiments and a PD mouse model for in vivo validation to study the pathophysiological mechanisms underneath PD-associated peritoneal fibrosis. High-glucose PD solution (Dianeal 4.25%, Baxter) increased protein expression of mesothelial-mesenchymal transition (MMT) markers, such as N-cadherin and α-SMA in MeT-5A cells, whereas it decreased catalase expression and stimulated the production of reactive oxygen species (ROS). Furthermore, macrophage influx and increased serum pro-inflammatory cytokines, such as IL-1β, MCP-1, and TNF-α, were observed in the PD mouse model. Interestingly, we discovered that oligo-fucoidan, an oligosaccharide extract from brown seaweed, successfully prevented PD-associated peritoneal thickening and fibrosis through antioxidant effect, downregulation of MMT markers, and attenuation of peritoneal and systemic inflammation. Hence, oligo-fucoidan has the potential to be developed into a novel preventive strategy for PD-associated peritoneal fibrosis.

Keywords: MMT; fibrosis; mesothelial–mesenchymal transition; oligo-fucoidan; peritoneal dialysis.

MeSH terms

  • Animals
  • Antioxidants / pharmacology
  • Cell Line
  • Cytokines / metabolism
  • Dialysis Solutions / chemistry
  • Dialysis Solutions / pharmacology
  • Disease Models, Animal*
  • Epithelial-Mesenchymal Transition / drug effects
  • Glucose / metabolism
  • Humans
  • Male
  • Mice
  • Mice, Inbred C57BL
  • Oligosaccharides / pharmacology
  • Peritoneal Dialysis* / adverse effects
  • Peritoneal Fibrosis* / drug therapy
  • Peritoneal Fibrosis* / prevention & control
  • Peritoneum / drug effects
  • Peritoneum / pathology
  • Reactive Oxygen Species / metabolism
  • Seaweed / chemistry

Substances

  • Reactive Oxygen Species
  • Cytokines
  • Antioxidants
  • Oligosaccharides
  • Glucose
  • Dialysis Solutions