[Alkaloid compounds in Nelumbinis Folium and their hypolipidemic effect]

Zhongguo Zhong Yao Za Zhi. 2024 Oct;49(19):5238-5243. doi: 10.19540/j.cnki.cjcmm.20240626.201.
[Article in Chinese]

Abstract

Four alkaloid compounds including one new compound and three known ones were isolated and extracted from the 70% ethanol extract of Nelumbinis Folium by silica gel column chromatography, octadecylsilyl(ODS) column chromatography and preparative high-performance liquid chromatography. Their structures were identified by nuclear magnetic resonance spectroscopy, high-resolution mass spectrometry, circular dichroism and other methods. Compound 1 was identified as a new compound and named as lotustine B(1). Compounds 2-4 were identified as nuciferin(2), dehydronuciferine(3), N-methylasimilobine(4). The effects of four isolated alkaloid compounds on total cholesterol(TC) and total triglycerides(TG) levels were evaluated by constructing a human hepatoma(HepG2) cell model of hyperlipidemia. The hypolipidemic effects of compounds 1-4 were also evaluated using oil red O staining experi-ments. The results showed that compound 4 can reduce the lipid levels of HepG2 cells and has potential hypolipidemic effects.

Keywords: Nelumbinis Folium; alkaloid compounds; hypolipidemic effect.

Publication types

  • English Abstract

MeSH terms

  • Alkaloids* / chemistry
  • Alkaloids* / pharmacology
  • Cholesterol
  • Drugs, Chinese Herbal* / chemistry
  • Drugs, Chinese Herbal* / pharmacology
  • Hep G2 Cells
  • Humans
  • Hyperlipidemias / drug therapy
  • Hypolipidemic Agents* / chemistry
  • Hypolipidemic Agents* / pharmacology
  • Molecular Structure
  • Nelumbo* / chemistry
  • Triglycerides / metabolism

Substances

  • Hypolipidemic Agents
  • Drugs, Chinese Herbal
  • Alkaloids
  • Triglycerides
  • Cholesterol