miR-21-5p Enriched Exosomes from Human Embryonic Stem Cells Promote Osteogenesis via YAP1 Modulation

Int J Nanomedicine. 2024 Dec 6:19:13095-13112. doi: 10.2147/IJN.S484751. eCollection 2024.

Abstract

Purpose: To investigate the osteogenic potential of human embryonic stem cell-derived exosomes (hESC-Exos) and their effects on the differentiation of human umbilical cord mesenchymal stem cells (hUCMSCs).

Methods: hESC-Exos were isolated and characterized using transmission electron microscopy (TEM), nanoparticle tracking analysis (NTA), and Western blotting. hUCMSCs were cultured with hESC-Exos to assess osteogenic differentiation through alizarin red staining, quantitative PCR (qPCR), and Western blotting. miRNA profiling of hESC-Exos was performed using miRNA microarray analysis. In vivo bone regeneration was evaluated using an ovariectomized rat model with bone defects treated with exosome-loaded scaffolds.

Results: hESC-Exos significantly promoted the osteogenic differentiation of hUCMSCs, as evidenced by increased alizarin red staining and the upregulation of osteogenesis-related genes and proteins (ALP, RUNX2, OCN). miRNA analysis revealed that miR-21-5p is a key regulator that targets YAP1 and activates the Wnt/β-catenin signaling pathway. In vivo, hESC-Exos enhanced bone repair in ovariectomized rats, as demonstrated by increased bone mineral density and improved bone microarchitecture compared to those in controls.

Conclusion: hESC-Exos exhibit significant osteogenic potential by promoting the differentiation of hUCMSCs and enhancing bone regeneration in vivo. This study revealed that the miR-21-5p-YAP1/β-catenin axis is a critical pathway, suggesting that the use of hESC-Exos is a promising therapeutic strategy for bone regeneration and repair.

Keywords: YAP1; bone regeneration; exosomes; human embryonic stem cells; miR-21-5p; osteogenic differentiation.

MeSH terms

  • Adaptor Proteins, Signal Transducing* / genetics
  • Adaptor Proteins, Signal Transducing* / metabolism
  • Animals
  • Bone Regeneration*
  • Cell Differentiation*
  • Cells, Cultured
  • Exosomes* / metabolism
  • Female
  • Human Embryonic Stem Cells* / cytology
  • Human Embryonic Stem Cells* / metabolism
  • Humans
  • Mesenchymal Stem Cells* / cytology
  • Mesenchymal Stem Cells* / metabolism
  • MicroRNAs* / genetics
  • Osteogenesis* / genetics
  • Osteogenesis* / physiology
  • Ovariectomy
  • Rats
  • Rats, Sprague-Dawley
  • Transcription Factors* / genetics
  • Transcription Factors* / metabolism
  • Wnt Signaling Pathway
  • YAP-Signaling Proteins*

Substances

  • MicroRNAs
  • YAP-Signaling Proteins
  • YAP1 protein, human
  • Transcription Factors
  • Adaptor Proteins, Signal Transducing
  • MIRN21 microRNA, human