SHIV remission in macaques with early treatment initiation and ultra long-lasting antiviral activity

Nat Commun. 2024 Dec 4;15(1):10550. doi: 10.1038/s41467-024-54783-0.

Abstract

Studies in SIV-infected macaques show that the virus reservoir is particularly refractory to conventional suppressive antiretroviral therapy (ART). We posit that optimized ART regimens designed to have robust penetration in tissue reservoirs and long-lasting antiviral activity may be advantageous for HIV or SIV remission. Here we treat macaques infected with RT-SHIV with oral emtricitabine/tenofovir alafenamide and long-acting cabotegravir/rilpivirine without (n = 4) or with (n = 4) the immune activator vesatolimod after the initial onset of viremia. We document full suppression in all animals during treatment (4-12 months) and no virus rebound after treatment discontinuation (1.5-2 years of follow up) despite CD8 + T cell depletion. We show efficient multidrug penetration in virus reservoirs and persisting rilpivirine in plasma for 2 years after the last dose. Our results document a type of virus remission that is achieved through early treatment initiation and provision of ultra long-lasting antiviral activity that persists after treatment cessation.

MeSH terms

  • Animals
  • Antiviral Agents* / administration & dosage
  • Antiviral Agents* / pharmacology
  • Antiviral Agents* / therapeutic use
  • CD8-Positive T-Lymphocytes / drug effects
  • CD8-Positive T-Lymphocytes / immunology
  • Diketopiperazines
  • Emtricitabine / administration & dosage
  • Emtricitabine / pharmacology
  • Emtricitabine / therapeutic use
  • Macaca mulatta
  • Male
  • Organophosphates / administration & dosage
  • Organophosphates / pharmacology
  • Organophosphates / therapeutic use
  • Pteridines
  • Pyridones / pharmacology
  • Simian Acquired Immunodeficiency Syndrome* / drug therapy
  • Simian Acquired Immunodeficiency Syndrome* / immunology
  • Simian Acquired Immunodeficiency Syndrome* / virology
  • Simian Immunodeficiency Virus* / drug effects
  • Simian Immunodeficiency Virus* / physiology
  • Tenofovir / administration & dosage
  • Tenofovir / pharmacology
  • Tenofovir / therapeutic use
  • Viral Load / drug effects
  • Viremia / drug therapy
  • Viremia / virology

Substances

  • Antiviral Agents
  • Emtricitabine
  • Tenofovir
  • vesatolimod
  • cabotegravir
  • Organophosphates
  • Pyridones
  • Pteridines
  • Diketopiperazines