Modafinil Versus Amphetamine-Dextroamphetamine For Idiopathic Hypersomnia and Narcolepsy Type 2: A Randomized, Blinded, Non-inferiority Trial

CNS Drugs. 2024 Nov;38(11):909-920. doi: 10.1007/s40263-024-01122-y. Epub 2024 Sep 21.

Abstract

Background and objective: Although there are several treatments for narcolepsy type 2 and idiopathic hypersomnia, studies that assess amphetamines, symptoms beyond sleepiness, and comparative effectiveness are needed. We performed a randomized, fully blinded, noninferiority trial of modafinil versus amphetamine-dextroamphetamine in these disorders.

Methods: Forty-four adults were randomized to modafinil or amphetamine-dextroamphetamine, individually titrated to a maximum of modafinil 200 mg twice daily or amphetamine-dextroamphetamine 20 mg twice daily, for 12 weeks. Primary outcome was change in Epworth from baseline to week 12, with a noninferiority threshold of 2 points. Secondary outcomes were (1) patient global impression of change measures of disease severity, sleepiness, sleep inertia, and cognition; (2) change from baseline in Hypersomnia Severity Index; and (3) change from baseline in Sleep Inertia Questionnaire. Adverse events were compared between groups.

Results: Epworth improved 5.0 [± standard deviation (SD) 2.7] points with modafinil and 4.4 (± SD 4.7) with amphetamine-dextroamphetamine; noninferiority of amphetamine-dextroamphetamine was not demonstrated (P = 0.11). Noninferiority of amphetamine-dextroamphetamine was demonstrated for change scores of severity, sleepiness, sleep inertia, Hypersomnia Severity Index, and Sleep Inertia Questionnaire. Dropouts due to adverse events were 31.8% for modafinil (including two severe events) and 9.1% for amphetamine-dextroamphetamine, P = 0.13. Anxiety was more common with modafinil and appetite suppression with amphetamine-dextroamphetamine.

Conclusion: Noninferiority of amphetamine-dextroamphetamine to modafinil was not demonstrated for the primary outcome. However, amphetamine-dextroamphetamine was noninferior on multiple secondary measures of disease severity and symptomatology. These data may inform shared decision-making regarding treatment for idiopathic hypersomnia and narcolepsy type 2.

Registration: Clinicaltrials.gov Registration (NCT03772314) 12/10/18. .

Publication types

  • Randomized Controlled Trial
  • Comparative Study

MeSH terms

  • Adult
  • Amphetamine / administration & dosage
  • Amphetamine / adverse effects
  • Benzhydryl Compounds / administration & dosage
  • Benzhydryl Compounds / adverse effects
  • Benzhydryl Compounds / pharmacology
  • Benzhydryl Compounds / therapeutic use
  • Central Nervous System Stimulants* / administration & dosage
  • Central Nervous System Stimulants* / adverse effects
  • Central Nervous System Stimulants* / therapeutic use
  • Dextroamphetamine* / administration & dosage
  • Dextroamphetamine* / adverse effects
  • Dextroamphetamine* / therapeutic use
  • Double-Blind Method
  • Female
  • Humans
  • Idiopathic Hypersomnia / diagnosis
  • Idiopathic Hypersomnia / drug therapy
  • Male
  • Middle Aged
  • Modafinil* / administration & dosage
  • Modafinil* / pharmacology
  • Modafinil* / therapeutic use
  • Narcolepsy* / drug therapy
  • Severity of Illness Index
  • Treatment Outcome
  • Wakefulness-Promoting Agents / administration & dosage
  • Wakefulness-Promoting Agents / pharmacology
  • Wakefulness-Promoting Agents / therapeutic use
  • Young Adult

Substances

  • Modafinil
  • Dextroamphetamine
  • Central Nervous System Stimulants
  • Benzhydryl Compounds
  • Wakefulness-Promoting Agents
  • Amphetamine

Associated data

  • ClinicalTrials.gov/NCT03772314