One Pot Synthesis of C3-Sulfurized Imidazolo [1,2- a] Pyridines

J Org Chem. 2024 Oct 4;89(19):14098-14107. doi: 10.1021/acs.joc.4c01524. Epub 2024 Sep 18.

Abstract

A facile and efficient annulation strategy was developed from easily accessible a-bromoketones, aminopyridines and benzazol, which afforded a series of imidazole [1,2-a]pyridine sulfides in moderate to good yields. The reaction involves the formation of C-N/C-S bond with the advantages of easy operation and wide substrates scope.