Identification of the forms of cytochrome P-450 induced in rat liver by 2-acetylaminofluorene using immunoblotting and partial purification

Biochem Biophys Res Commun. 1985 Apr 30;128(2):578-85. doi: 10.1016/0006-291x(85)90085-3.

Abstract

The amounts of 5 different forms of cytochrome P-450 in liver microsomes from rats treated with 2-acetylaminofluorene were determined and compared with the corresponding patterns in microsomes from control, 3-methylcholanthrene- and phenobarbital-treated animals. 2-Acetylaminofluorene was found to increase the amount of cytochromes P-450b + e 10-fold and of cytochrome P-450d 3-fold, while there was a 54% increase in the level of cytochrome P-450 PB/PCN-E. Cytochrome P-450c was increased from a level too low to detect (less than 0.001 pmol/mg protein) to 0.019 pmol/mg protein. These findings were also confirmed by partial purification of cytochromes P-450b + e and c after 2-acetylaminofluorene treatment.

Publication types

  • Research Support, Non-U.S. Gov't
  • Research Support, U.S. Gov't, P.H.S.

MeSH terms

  • 2-Acetylaminofluorene / pharmacology*
  • Animals
  • Cytochrome P-450 Enzyme System / biosynthesis*
  • Enzyme Induction
  • Immunosorbent Techniques
  • Isoenzymes / biosynthesis*
  • Male
  • Methylcholanthrene / pharmacology
  • Microsomes, Liver / drug effects
  • Microsomes, Liver / enzymology*
  • Phenobarbital / pharmacology
  • Rats
  • Rats, Inbred Strains

Substances

  • Isoenzymes
  • Methylcholanthrene
  • Cytochrome P-450 Enzyme System
  • 2-Acetylaminofluorene
  • Phenobarbital