Comparison of thrombogenicity in different types of drug-eluting stents during transition from DAPT to SAPT

Catheter Cardiovasc Interv. 2024 Jul;104(1):10-20. doi: 10.1002/ccd.31083. Epub 2024 May 20.

Abstract

Background: During the transition from dual antiplatelet therapy (DAPT) to single antiplatelet therapy (SAPT), previous studies have raised concerns about a rebound effect. We compared platelet and inflammatory cell adhesion on different types of stents in the setting of clopidogrel presence and withdrawal.

Methods: In Experiment 1, three pigs were administered with DAPT, that is, clopidogrel and acetylsalicylic acid (ASA), for 7 days. Each animal underwent an extracorporeal carotid arteriovenous shunt model implanted with fluoropolymer-coated everolimus-eluting stent (FP-EES), biodegradable-polymer sirolimus-eluting stent (BP-SES), and biodegradable-polymer everolimus-eluting stents (BP-EES). In Experiment 2, two pigs were administered DAPT, clopidogrel was then withdrawn at day 7, and SAPT with ASA was continued for next 21 days. Then flow-loop experiments with the drawn blood from each time point were performed for FP-EES, BioLinx-polymer zotarolimus-eluting stents (BL-ZES), and BP-EES. The rebound effect was defined as the statistical increase of inflammation and platelet adhesion assessed with immunohistochemistry on the stent-strut level basis from baseline to day-14 or 28.

Results: Both experiments showed platelet adhesion value was highest in BP-EES, while the least in FP-EES during DAPT therapy. There was no increase in platelet or inflammatory cell adhesion above baseline values (i.e., no therapy) due to the cessation of clopidogrel on the stent-strut level. Monocyte adhesion was the least for FP-EES with the same trend observed for neutrophil adhesion.

Conclusions: No evidence of rebound effect was seen after the transition from DAPT to SAPT. FP-EES demonstrated the most favorable antithrombotic and anti-inflammatory profile regardless of the different experimental designs.

Keywords: coronary artery disease; drug‐eluting stent; dual antiplatelet therapy; rebound effect; single antiplatelet therapy.

Publication types

  • Comparative Study

MeSH terms

  • Animals
  • Arteriovenous Shunt, Surgical / adverse effects
  • Aspirin* / administration & dosage
  • Blood Platelets / drug effects
  • Blood Platelets / metabolism
  • Clopidogrel* / administration & dosage
  • Clopidogrel* / pharmacology
  • Disease Models, Animal
  • Drug Administration Schedule
  • Drug-Eluting Stents*
  • Dual Anti-Platelet Therapy*
  • Everolimus* / administration & dosage
  • Everolimus* / pharmacology
  • Platelet Adhesiveness* / drug effects
  • Platelet Aggregation Inhibitors* / administration & dosage
  • Platelet Aggregation Inhibitors* / adverse effects
  • Platelet Aggregation Inhibitors* / pharmacology
  • Prosthesis Design*
  • Sirolimus* / administration & dosage
  • Sirolimus* / analogs & derivatives
  • Sirolimus* / pharmacology
  • Sus scrofa
  • Thrombosis* / etiology
  • Thrombosis* / prevention & control
  • Time Factors

Substances

  • Platelet Aggregation Inhibitors
  • Clopidogrel
  • Sirolimus
  • Everolimus
  • Aspirin
  • zotarolimus