Antagonism of let-7c reduces atherosclerosis and macrophage lipid accumulation by promoting PGC-1α/LXRα/ABCA1/G1 pathway

Gene. 2024 May 30:909:148302. doi: 10.1016/j.gene.2024.148302. Epub 2024 Feb 23.

Abstract

Changes in circulating let-7c were significantly associated with the alter in lipid profile, but its role in intracellular lipid metabolism remains unknown. This work was conducted to explore the effects of let-7c on the lipid accumulation in macrophages and uncover the underlying mechanism. Our results showed that let-7c inhibition relieved atherosclerosis progression in apoE-/- mice. In ox-LDL-treatment macrophages, let-7c knockdown suppressed lipid accumulation but does no affect cholesterol intake. Consistent with this, overexpression of let-7c promoted lipid accumulation by reducing the expression of LXRα and ABCA1/G1. Mechanistically, let-7c targeted PGC-1α to repress the expression of LXRα and ABCA1/G1, thereby regulating cholesterol homeostasis in macrophages. Taken together, these findings suggest that antagonism of let-7c reduces atherosclerosis and macrophage lipid accumulation through the PGC-1α/LXRα/ABCA1/G1 axis.

Keywords: ABCA/G1; Atherosclerosis; Cholesterol homeostasis; Macrophages; MicroRNAs.

MeSH terms

  • ATP Binding Cassette Transporter 1 / genetics
  • ATP Binding Cassette Transporter 1 / metabolism
  • Animals
  • Atherosclerosis* / genetics
  • Atherosclerosis* / metabolism
  • Cholesterol / metabolism
  • Hypercholesterolemia* / metabolism
  • Lipid Metabolism / genetics
  • Liver X Receptors / genetics
  • Liver X Receptors / metabolism
  • Macrophages / metabolism
  • Mice

Substances

  • Cholesterol
  • ATP Binding Cassette Transporter 1
  • Liver X Receptors