Perspectives on Ensifentrine and Its Therapeutic Potential in the Treatment of COPD: Evidence to Date

Int J Chron Obstruct Pulmon Dis. 2024 Jan 3:19:11-16. doi: 10.2147/COPD.S385811. eCollection 2024.

Abstract

Ensifentrine is a novel inhalational phosphodiesterase (PDE)3 and PDE4 inhibitor which improves bronchodilation and decreases inflammatory markers by acting locally on the bronchial tissue, with minimal systemic effects. Both preclinical and clinical trials have demonstrated benefits of this therapy, including improvement in lung function and reduction in exacerbations. This therapy is currently under review by the US Food and Drug Administration with a decision expected in 2024.

Keywords: chronic obstructive pulmonary disease; phosphodiesterase inhibitor; therapy.

Publication types

  • Review

MeSH terms

  • Bronchi
  • Humans
  • Isoquinolines
  • Pulmonary Disease, Chronic Obstructive* / diagnosis
  • Pulmonary Disease, Chronic Obstructive* / drug therapy
  • Pyrimidinones
  • United States

Substances

  • ensifentrine
  • Isoquinolines
  • Pyrimidinones