Structure and Dynamics Guiding Design of Antibody Therapeutics and Vaccines

Antibodies (Basel). 2023 Oct 18;12(4):67. doi: 10.3390/antib12040067.

Abstract

Antibodies and other new antibody-like formats have emerged as one of the most rapidly growing classes of biotherapeutic proteins. Understanding the structural features that drive antibody function and, consequently, their molecular recognition is critical for engineering antibodies. Here, we present the structural architecture of conventional IgG antibodies alongside other formats. We emphasize the importance of considering antibodies as conformational ensembles in solution instead of focusing on single-static structures because their functions and properties are strongly governed by their dynamic nature. Thus, in this review, we provide an overview of the unique structural and dynamic characteristics of antibodies with respect to their antigen recognition, biophysical properties, and effector functions. We highlight the numerous technical advances in antibody structure prediction and design, enabled by the vast number of experimentally determined high-quality structures recorded with cryo-EM, NMR, and X-ray crystallography. Lastly, we assess antibody and vaccine design strategies in the context of structure and dynamics.

Keywords: NMR; X-ray crystallography; antibody; antibody structure determination; cryo-EM; molecular dynamics; special formats; structure prediction; vaccine design.

Publication types

  • Review

Grants and funding

N.D.P. has received funding from the European Union’s Horizon 2020 research and innovation program under the Marie Skłodowska-Curie grant agreement number 847476. The views and opinions expressed herein do not necessarily reflect those of the European Commission. This work was supported by the Austrian Science Fund (FWF) via grant P34518. This work was supported by the Austrian Academy of Sciences APART-MINT postdoctoral fellowship to M.L.F.Q. H.R.P. was supported by a David C. Fairchild Endowed Fellowship, and the Achievement Rewards for College Scientists Foundation. J.H, J.F. and A.B.W. were supported by the Bill and Melinda Gates Foundation through grant INV-004923 (A.B.W.).