Extended-release tacrolimus dosing and outcomes in pediatric and young adult transplant recipients - A single-center experience

Pediatr Transplant. 2024 Feb;28(1):e14611. doi: 10.1111/petr.14611. Epub 2023 Sep 21.

Abstract

Background: Published data on LCP-tacrolimus (LCPT) in the pediatric population are limited.

Methods: This single-center, retrospective, observational study describes LCPT doses needed to reach therapeutic ranges in pediatric and young adult kidney and liver transplant recipients in both de novo usage and conversion from immediate-release tacrolimus (IR-Tac). Adverse outcomes up to 12 months after LCPT initiation were also evaluated.

Results: Forty-one transplant recipients (30 kidney, 11 liver) were included. The median initial doses of LCPT were 0.034 mg/kg (IQR 0.019) de novo and 0.09 mg/kg (IQR = 0.076) converted. The median doses at first therapeutic level were 0.086 mg/kg (IQR 0.028) de novo and 0.1 mg/kg (IQR 0.066) converted. The median LCPT:IR-Tac conversion ratio initially was 0.7 and 0.75 at therapeutic levels. The rate of AKI per 100 days of exposure to IR-Tac was 0.546 and 0.439 on LCPT. The percentage of patients with rejection was not different before and after conversion (clinical rejection 8.6% [n = 3] vs 11.4% [n = 4], p = .6; biopsy-proven rejection 2.9% [n = 1] vs 11.4% [n = 4], p = .11). One patient had graft loss unrelated to rejection, and the graft was explanted.

Conclusion: In this study, pediatric and young adult abdominal transplant recipients had therapeutic tacrolimus levels at LCPT doses below the adult-labeled dose; the conversion ratio from IR-Tac to LCPT at therapeutic level was similar. There were no identified safety concerns in de novo or converted LCPT use in pediatric and young adult patients.

Keywords: extended-release tacrolimus; kidney transplant; liver transplant; pediatric.

Publication types

  • Observational Study

MeSH terms

  • Child
  • Drug Administration Schedule
  • Graft Rejection / drug therapy
  • Graft Rejection / prevention & control
  • Humans
  • Immunosuppressive Agents / adverse effects
  • Kidney Transplantation* / adverse effects
  • Prospective Studies
  • Tacrolimus*
  • Transplant Recipients
  • Young Adult

Substances

  • Tacrolimus
  • Immunosuppressive Agents