Leflunomide exposure through second trimester of pregnancy: A case report

Birth Defects Res. 2023 Oct 1;115(16):1566-1569. doi: 10.1002/bdr2.2221. Epub 2023 Jul 18.

Abstract

Leflunomide is a commonly used disease modifying antirheumatic agent. However, its use is contraindicated in pregnancy. The American College of Rheumatology (ACR) guidelines recommend discontinuing Leflunomide at least 24 months before conception. If a woman is found to be pregnant while on Leflunomide, ACR suggests close monitoring and cholestyramine washout. We describe a case of a patient with a history of juvenile idiopathic arthritis who was on Leflunomide throughout the first and second trimester of her pregnancy. A cholestyramine washout regimen was started but not completed. The patient was induced at 37 weeks of gestation due to non-reassuring fetal heart rate. She ultimately delivered a healthy baby via emergency cesarian section.

Keywords: Leflunomide; pregnancy; rheumatoid arthritis; teratogen.

Publication types

  • Case Reports

MeSH terms

  • Arthritis, Rheumatoid*
  • Cholestyramine Resin*
  • Female
  • Humans
  • Isoxazoles / adverse effects
  • Leflunomide
  • Pregnancy
  • Pregnancy Trimester, Second

Substances

  • Leflunomide
  • Cholestyramine Resin
  • Isoxazoles