Influence of indomethacin on an increase in cerebral blood flow induced by KC-404, a novel cerebral vasodilator, in an anesthetized dog

Gen Pharmacol. 1986;17(3):339-41. doi: 10.1016/0306-3623(86)90050-9.

Abstract

The effect of KC-404 on vertebral blood flow in the absence and presence of indomethacin was investigated in an anesthetized dog. KC-404 (0.2 mg/kg, i.v.) showed a significant and long lasting increase in vertebral blood flow. This was markedly diminished by pretreatment of the animal with indomethacin. The increase in heart rate due to KC-404 administration was also diminished, though moderately, by pretreatment with indomethacin. From these results, the possible mechanism of action of KC-404 was discussed, particularly in reference to cerebral vasodilating prostaglandins.

MeSH terms

  • Animals
  • Cerebrovascular Circulation / drug effects*
  • Dogs
  • Female
  • Hemodynamics / drug effects
  • Indomethacin / pharmacology*
  • Male
  • Pyridines / antagonists & inhibitors*
  • Pyridines / pharmacology
  • Vasodilator Agents / antagonists & inhibitors*
  • Vasodilator Agents / pharmacology
  • Vertebral Artery

Substances

  • Pyridines
  • Vasodilator Agents
  • ibudilast
  • Indomethacin