Evaluation of triacontanol-containing compounds as anti-inflammatory agents using guinea pig models

J Invest Dermatol. 1987 Oct;89(4):380-3. doi: 10.1111/1523-1747.ep12471763.

Abstract

A mixture of the aliphatic alcohol, triacontanol, and other chemically associated naturally occurring alcohols was applied to the denuded dorsal cutaneous surface of guinea pigs to evaluate anti-inflammatory activity. In the setting of a chemical irritation with 2% croton oil and in an allergic dermatitis created with dinitrochlorobenzene sensitization and challenge, the triacontanol-containing preparation was significantly more effective than vehicle alone (DHL skin cream) but not as effective as 0.05% Diprolene ointment. Lymphocyte stimulation was studied by tritiated thymidine uptake and morphologic examination for blast transformation. When triacontanol-containing compounds were solubilized in aqueous media, effects on lymphocytes were insignificant. When solubilized in ethanol, there was a marked effect on thymidine uptake but not on blast transformation when compared to parallel controls.

MeSH terms

  • Animals
  • Anti-Inflammatory Agents*
  • Betamethasone / analogs & derivatives*
  • Betamethasone / pharmacology
  • Betamethasone / therapeutic use
  • Dermatitis, Contact / drug therapy
  • Fatty Alcohols / pharmacology*
  • Fatty Alcohols / therapeutic use
  • Guinea Pigs
  • Lymphocyte Activation / drug effects

Substances

  • Anti-Inflammatory Agents
  • Fatty Alcohols
  • 1-triacontanol
  • betamethasone-17,21-dipropionate
  • Betamethasone