Changing Surface Polyethylene Glycol Architecture Affects Elongated Nanoparticle Penetration into Multicellular Tumor Spheroids

Biomacromolecules. 2022 Aug 8;23(8):3296-3307. doi: 10.1021/acs.biomac.2c00386. Epub 2022 Jul 11.

Abstract

Nanoparticles (NPs) designed for biomedical applications are coated with protein-repellent polymers. Here, we examine the penetration of rodlike NPs with narrow size distributions (Ln = 170 nm, wn = 12 nm) into multicellular tumor spheroids prepared from two human cancer cell lines. Two types of NPs with different core materials [polyferrocenylsilane and cellulose nanocrystals (CNC)] were coated with a dense brush of poly(oligoethyleneglycol methacrylate) (POEGMA), while a second CNC NP sample was coated with a linear polyethylene glycol (PEG) brush. While the core material had little influence, the coating material was strikingly important, with POEGMA-coated NPs penetrating much more deeply into the tumor spheroids than the NPs coated with linear PEG. Localization experiments using 111In-labeled POEGMA-coated CNC NPs showed that most of the radioactivity remained in the interstitial space (ca. 78%) with little cell uptake (ca. 6%). Hence, the deep penetration of these nanorods into tumor spheroids is associated with an interstitial diffusion pathway through the extracellular matrix and not cellular transcytosis.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Humans
  • Nanoparticles* / chemistry
  • Neoplasms* / drug therapy
  • Neoplasms* / metabolism
  • Particle Size
  • Polyethylene Glycols / chemistry
  • Spheroids, Cellular / metabolism

Substances

  • Polyethylene Glycols