Effects of fluocinolone acetonide on mouse skin sterol metabolism and two-stage carcinogenesis

Carcinogenesis. 1988 Sep;9(9):1661-4. doi: 10.1093/carcin/9.9.1661.

Abstract

Fluocinolone acetonide (FA) is one of the most potent synthetic glucocorticoids and is known to possess an anti-tumor promoting activity. An attempt was made to evaluate this activity by estimating tumor promoting activity. Unexpectedly, when 10 micrograms of FA was applied alone or after a single application of a subcarcinogenic dose of 3-methylcholanthrene to mouse skin, results suggested that FA itself may be a tumor promoter or a complete carcinogen. Other glucocorticoids tested, e.g. dexamethasone, hydrocortisone and prednisolone, also revealed similar effects but were less potent than FA. To verify the possibility that glucocorticoid is a complete carcinogen or a tumor promoter, a tumor incidence experiment was performed for 24 weeks. As a result it was found that FA possesses a tumor promoting activity at some dose levels but no tumor initiating activity.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Animals
  • Chromatography, Gas
  • Dose-Response Relationship, Drug
  • Fluocinolone Acetonide / pharmacology*
  • Methylcholanthrene / pharmacology
  • Mice
  • Skin / metabolism*
  • Skin Neoplasms / chemically induced*
  • Skin Neoplasms / metabolism
  • Sterols / metabolism*
  • Tetradecanoylphorbol Acetate / pharmacology

Substances

  • Sterols
  • Fluocinolone Acetonide
  • Methylcholanthrene
  • Tetradecanoylphorbol Acetate