Role of host factors in SARS-CoV-2 entry

J Biol Chem. 2021 Jul;297(1):100847. doi: 10.1016/j.jbc.2021.100847. Epub 2021 May 28.

Abstract

The zoonotic transmission of highly pathogenic coronaviruses into the human population is a pressing concern highlighted by the ongoing SARS-CoV-2 pandemic. Recent work has helped to illuminate much about the mechanisms of SARS-CoV-2 entry into the cell, which determines host- and tissue-specific tropism, pathogenicity, and zoonotic transmission. Here we discuss current findings on the factors governing SARS-CoV-2 entry. We first reviewed key features of the viral spike protein (S) mediating fusion of the viral envelope and host cell membrane through binding to the SARS-CoV-2 receptor, angiotensin-converting enzyme 2. We then examined the roles of host proteases including transmembrane protease serine 2 and cathepsins in processing S for virus entry and the impact of this processing on endosomal and plasma membrane virus entry routes. We further discussed recent work on several host cofactors that enhance SARS-CoV-2 entry including Neuropilin-1, CD147, phosphatidylserine receptors, heparan sulfate proteoglycans, sialic acids, and C-type lectins. Finally, we discussed two key host restriction factors, i.e., interferon-induced transmembrane proteins and lymphocyte antigen 6 complex locus E, which can disrupt SARS-CoV-2 entry. The features of SARS-CoV-2 are presented in the context of other human coronaviruses, highlighting unique aspects. In addition, we identify the gaps in understanding of SARS-CoV-2 entry that will need to be addressed by future studies.

Keywords: ACE2; RNA virus; SARS-CoV-2; TMPRSS2; cathepsin B; endocytosis; entry cofactor; membrane fusion; virus entry; virus receptor.

Publication types

  • Research Support, N.I.H., Extramural
  • Review

MeSH terms

  • Animals
  • Basigin / genetics
  • Basigin / metabolism
  • COVID-19 / genetics
  • COVID-19 / metabolism*
  • COVID-19 / virology
  • Host-Pathogen Interactions
  • Humans
  • Lectins, C-Type / genetics
  • Lectins, C-Type / metabolism
  • Neuropilin-1 / genetics
  • Neuropilin-1 / metabolism
  • Receptors, Virus / genetics
  • Receptors, Virus / metabolism
  • SARS-CoV-2 / genetics
  • SARS-CoV-2 / physiology*
  • Virus Internalization*

Substances

  • Lectins, C-Type
  • Receptors, Virus
  • Basigin
  • Neuropilin-1