Safety of nelarabine in adults with relapsed or refractory T-cell acute lymphoblastic leukemia/lymphoma

Expert Opin Drug Saf. 2021 Jul;20(7):751-756. doi: 10.1080/14740338.2021.1919621. Epub 2021 May 17.

Abstract

Introduction: T-cell acute lymphoblastic leukemia (T-ALL) and lymphoma (T-LBL) are aggressive hematological malignancies accounting for 15-20% of adult acute lymphoproliferative diseases. Treatment of relapsed/refractory (R/R) T-ALL/T-LBL is challenging with very few therapeutic options.

Areas covered: This report provides a concise review on the efficacy and safety of nelarabine monotherapy in adults with R/R T-ALL and T-LBL.

Expert opinion: Nelarabine is approved for the treatment of adults with R/R T-ALL/T-LBL in the setting of third or more line of therapy. Hematological and neurological toxicities are the most frequent adverse events. Grade 3 and 4 neutropenia and thrombocytopenia are common, however with treatment-related deaths accounting only for 1-2% of patients. Neurological toxicity is typically characterized by a reversible peripheral neuropathy, usually mild or moderate and without treatment delay. Other neurological (somnolence and depressed level of consciousness) or extra-neurological adverse events are uncommon and rarely severe. In conclusion, nelarabine is a well tolerated and effective salvage therapy in patients with R/R T-ALL/T-LBL and has acquired an important role as a bridge-therapy to allogeneic stem cell transplantation.

Keywords: Nelarabine; acute lymphoblastic leukemia; lymphoblastic lymphoma; neurotoxicity.

Publication types

  • Review

MeSH terms

  • Adult
  • Antineoplastic Agents / administration & dosage*
  • Antineoplastic Agents / adverse effects
  • Arabinonucleosides / administration & dosage*
  • Arabinonucleosides / adverse effects
  • Hematopoietic Stem Cell Transplantation
  • Humans
  • Precursor T-Cell Lymphoblastic Leukemia-Lymphoma / drug therapy*
  • Recurrence
  • Salvage Therapy

Substances

  • Antineoplastic Agents
  • Arabinonucleosides
  • nelarabine