Orally delivered MK-4482 inhibits SARS-CoV-2 replication in the Syrian hamster model

Nat Commun. 2021 Apr 16;12(1):2295. doi: 10.1038/s41467-021-22580-8.

Abstract

The COVID-19 pandemic progresses unabated in many regions of the world. An effective antiviral against SARS-CoV-2 that could be administered orally for use following high-risk exposure would be of substantial benefit in controlling the COVID-19 pandemic. Herein, we show that MK-4482, an orally administered nucleoside analog, inhibits SARS-CoV-2 replication in the Syrian hamster model. The inhibitory effect of MK-4482 on SARS-CoV-2 replication is observed in animals when the drug is administered either beginning 12 h before or 12 h following infection in a high-risk exposure model. These data support the potential utility of MK-4482 to control SARS-CoV-2 infection in humans following high-risk exposure as well as for treatment of COVID-19 patients.

Publication types

  • Research Support, N.I.H., Intramural
  • Research Support, Non-U.S. Gov't

MeSH terms

  • Administration, Oral
  • Animals
  • Antiviral Agents / administration & dosage*
  • COVID-19 / virology
  • COVID-19 Drug Treatment*
  • Chlorocebus aethiops
  • Cytidine / administration & dosage
  • Cytidine / analogs & derivatives*
  • Disease Models, Animal
  • Humans
  • Hydroxylamines / administration & dosage*
  • Mesocricetus
  • SARS-CoV-2 / drug effects*
  • SARS-CoV-2 / isolation & purification
  • SARS-CoV-2 / physiology
  • Vero Cells
  • Virus Replication / drug effects*

Substances

  • Antiviral Agents
  • Hydroxylamines
  • Cytidine
  • molnupiravir