Drug resistance in protozoan parasites

Emerg Top Life Sci. 2017 Dec 22;1(6):627-632. doi: 10.1042/ETLS20170113.

Abstract

As with all other anti-infectives (antibiotics, anti-viral drugs, and anthelminthics), the limited arsenal of anti-protozoal drugs is being depleted by a combination of two factors: increasing drug resistance and the failure to replace old and often shamefully inadequate drugs, including those compromised by (cross)-resistance, through the development of new anti-parasitics. Both factors are equally to blame: a leaking bathtub may have plenty of water if the tap is left open; if not, it will soon be empty. Here, I will reflect on the factors that contribute to the drug resistance emergency that is unfolding around us, specifically resistance in protozoan parasites.

Keywords: chemotherapy; drug resistance; drug transporter; multidrug resistance; parasitic protozoa; resistance mechanism.