Persistence of fluphenazine in plasma after decanoate withdrawal

J Clin Psychopharmacol. 1988 Feb;8(1):53-6.

Abstract

We discontinued fluphenazine decanoate using a double-blind, crossover random order design, in 12 recent onset clinically stable schizophrenics who had been given fluphenazine decanoate 12.5 mg intramuscularly every 2 weeks for at least 1 year prior to drug withdrawal. Each condition (drug or placebo) lasted 12 weeks. Using a radioimmunoassay verified by comparison to a gas chromatographic-mass spectrometric method, plasma fluphenazine levels were measured every 2 weeks during drug continuation and drug withdrawal conditions. No patient relapsed over the 24-week period of the study. Mean fluphenazine levels between drug continuation and withdrawal conditions showed a progressively larger difference over time, although significant differences were not seen until week 8. By week 12 after drug withdrawal, 33% of subjects still showed notable plasma fluphenazine levels. On the basis of our preliminary findings, we suggest that 2-week intervals between injections may be too short and that wider intervals may achieve similar clinical results.

Publication types

  • Clinical Trial
  • Randomized Controlled Trial
  • Research Support, Non-U.S. Gov't
  • Research Support, U.S. Gov't, P.H.S.

MeSH terms

  • Adult
  • Female
  • Fluphenazine / analogs & derivatives*
  • Fluphenazine / blood*
  • Fluphenazine / pharmacokinetics
  • Fluphenazine / therapeutic use
  • Humans
  • Male
  • Radioimmunoassay
  • Schizophrenia / drug therapy
  • Substance Withdrawal Syndrome / blood*

Substances

  • fluphenazine depot
  • Fluphenazine