Endoscopy-controlled study of the safety of nabumetone compared with naproxen in arthritis therapy

Am J Med. 1987 Oct 30;83(4B):25-30. doi: 10.1016/0002-9343(87)90589-4.

Abstract

Nonsteroidal anti-inflammatory drug (NSAID) gastropathy is now a commonly recognized and reported complication of such arthritis therapy. Significant gastric lesions develop in up to 40 percent of arthritic patients treated with long-term anti-inflammatory doses of NSAIDs, 20 percent of which represents actual ulcer crater disease. This 12-week endoscopy-controlled, double-blind study was constructed to evaluate the safety and efficacy of nabumetone 1,000 mg at bedtime compared with naproxen 250 mg twice daily. A total of 37 patients completed the study, including 29 patients with a diagnosis of osteoarthritis and eight with a diagnosis of rheumatoid arthritis. By posttreatment endoscopy, nabumetone was significantly less toxic to the gastrointestinal tract than was naproxen. The nabumetone-treated group also showed greater improvement in all efficacy variables, with significant improvement noted in three of these five variables in both rheumatoid and osteoarthritic patients.

Publication types

  • Clinical Trial
  • Comparative Study
  • Controlled Clinical Trial

MeSH terms

  • Adult
  • Aged
  • Anti-Inflammatory Agents, Non-Steroidal / adverse effects
  • Anti-Inflammatory Agents, Non-Steroidal / therapeutic use*
  • Arthritis, Rheumatoid / drug therapy*
  • Butanones / adverse effects
  • Butanones / therapeutic use*
  • Clinical Trials as Topic
  • Double-Blind Method
  • Duodenoscopy
  • Endoscopy*
  • Esophagoscopy
  • Female
  • Gastric Mucosa / drug effects
  • Gastric Mucosa / pathology
  • Gastroscopy
  • Humans
  • Male
  • Middle Aged
  • Nabumetone
  • Naproxen / adverse effects
  • Naproxen / therapeutic use*
  • Osteoarthritis / drug therapy*

Substances

  • Anti-Inflammatory Agents, Non-Steroidal
  • Butanones
  • Naproxen
  • Nabumetone