Avobenzone incorporation in a diverse range of Ru(II) scaffolds produces potent potential antineoplastic agents

Dalton Trans. 2020 Sep 15;49(35):12161-12167. doi: 10.1039/d0dt02016h.

Abstract

Four structurally distinct classes of polypyridyl ruthenium complexes containing avobenzone exhibited low micromolar and submicromolar potencies in cancer cells, and were up to 273-fold more active than the parent ligand. Visible light irradiation enhanced the cytotoxicity of some complexes, making them promising candidates for combined chemo-photodynamic therapy.

MeSH terms

  • Antineoplastic Agents / chemistry*
  • Antineoplastic Agents / pharmacology*
  • Cell Line, Tumor
  • Coordination Complexes / chemistry*
  • Coordination Complexes / pharmacology*
  • Humans
  • Ligands
  • Photochemotherapy
  • Propiophenones / chemistry*
  • Ruthenium / chemistry*
  • Structure-Activity Relationship

Substances

  • Antineoplastic Agents
  • Coordination Complexes
  • Ligands
  • Propiophenones
  • Ruthenium
  • avobenzone