Inspiratory neural drive and dyspnea in interstitial lung disease: Effect of inhaled fentanyl

Respir Physiol Neurobiol. 2020 Nov:282:103511. doi: 10.1016/j.resp.2020.103511. Epub 2020 Aug 3.

Abstract

Background: Exertional dyspnea in interstitial lung disease (ILD) remains difficult to manage despite advances in disease-targeted therapies. Pulmonary opioid receptors present a potential therapeutic target for nebulized fentanyl to provide dyspnea relief.

Methods: ILD patients were characterized with reference to healthy volunteers. A randomized, double-blind, placebo-controlled crossover comparison of 100 mcg nebulized fentanyl vs placebo on dyspnea intensity and inspiratory neural drive (IND) during constant work rate (CWR) cycle exercise was performed in 21 ILD patients.

Results: Dyspnea intensity in ILD increased in association with an increase in IND (diaphragm activation) from a high resting value of 16.66 ± 6.52 %-60.04 ± 12.52 % of maximum (r = 0.798, p < 0.001). At isotime during CWR exercise, Borg dyspnea intensity ratings with fentanyl vs placebo were 4.1 ± 1.2 vs 3.8 ± 1.2, respectively (p = 0.174), and IND responses were also similar.

Conclusion: IND rose sharply during constant work rate exercise in association with dyspnea intensity in mild to moderate ILD but was not different after nebulized fentanyl compared with placebo.

Keywords: Dyspnoea; Fentanyl; Interstitial lung disease; Nebulized treatment; Respiratory physiology.

Publication types

  • Randomized Controlled Trial
  • Research Support, Non-U.S. Gov't

MeSH terms

  • Administration, Inhalation
  • Aged
  • Aged, 80 and over
  • Analgesics, Opioid / administration & dosage
  • Analgesics, Opioid / pharmacology*
  • Cross-Over Studies
  • Diaphragm / physiopathology
  • Double-Blind Method
  • Dyspnea / drug therapy*
  • Dyspnea / etiology
  • Dyspnea / physiopathology*
  • Electromyography
  • Exercise / physiology*
  • Female
  • Fentanyl / administration & dosage
  • Fentanyl / pharmacology*
  • Humans
  • Inhalation / physiology*
  • Lung Diseases, Interstitial / complications
  • Lung Diseases, Interstitial / physiopathology*
  • Male
  • Middle Aged
  • Nebulizers and Vaporizers
  • Physical Exertion / physiology
  • Treatment Outcome

Substances

  • Analgesics, Opioid
  • Fentanyl