Antigenic contraction of guinea pig tracheal preparations passively sensitized with monoclonal IgE: pharmacological modulation

Int Arch Allergy Appl Immunol. 1988;87(4):342-8. doi: 10.1159/000234699.

Abstract

Spirally cut guinea pig tracheal preparations were passively sensitized using a mouse monoclonal IgE antibody against dinitrophenol (DNP). Maximal contraction observed following challenge with DNP-bovine serum albumin (DNP-BSA, 5 micrograms/ml; n = 20) response was approximately 46% of the histamine response (0.52 +/- 0.09 g/mm2; n = 53). Indomethacin (1.7 microM) increased and PGE2 (1 microM) decreased the response to the antigen. FPL 55712 (10 microM), atropine (0.1 microM), L 651392 (5 microM) or tripelennamine (1 microM) always reduced the maximal DNP-BSA response, but not BN 52021 (100 microM). This model may be used for rapid detection of compounds with antiallergic properties on IgE-dependent lung pathological states.

MeSH terms

  • Animals
  • Antibodies, Monoclonal / physiology*
  • Antigens / immunology*
  • Atropine / pharmacology
  • Chromones / pharmacology
  • Dinitrophenols / immunology*
  • Dose-Response Relationship, Immunologic
  • Guinea Pigs
  • Immunization, Passive*
  • Immunoglobulin E / physiology*
  • Male
  • Mice
  • Mice, Inbred BALB C
  • Muscle Contraction / drug effects*
  • Phenothiazines / pharmacology
  • Serum Albumin, Bovine / immunology*
  • Trachea
  • Tripelennamine / pharmacology

Substances

  • Antibodies, Monoclonal
  • Antigens
  • Chromones
  • Dinitrophenols
  • Phenothiazines
  • dinitrophenyl-bovine serum albumin
  • Serum Albumin, Bovine
  • Immunoglobulin E
  • Tripelennamine
  • Atropine
  • FPL 55712
  • 4-bromo-2,7-dimethoxy-3H-phenothiazin-3-one