Amphetamine-induced sensitization of hypertension and lamina terminalis neuroinflammation

Am J Physiol Regul Integr Comp Physiol. 2020 Mar 1;318(3):R649-R656. doi: 10.1152/ajpregu.00233.2019. Epub 2020 Feb 12.

Abstract

Psychomotor stimulants are prescribed for many medical conditions, including obesity, sleep disorders, and attention-deficit/hyperactivity disorder. However, despite their acknowledged therapeutic utility, these stimulants are frequently abused, and their use can have both short- and long-term negative consequences. Although stimulants such as amphetamines acutely elevate blood pressure, it is unclear whether they cause any long-term effects on cardiovascular function after use has been discontinued. Previous work in our laboratory has demonstrated that physiological and psychosocial stressors will produce sensitization of the hypertensive response, a heightened pressor response to a hypertensinogenic stimulus delivered after stressor exposure. Here, we tested whether pretreatment with amphetamine for 1 wk can sensitize the hypertensive response in rats. We found that repeated amphetamine administration induced and maintained sensitization of the pressor response to angiotensin II following a 7-day delay after amphetamine injections were terminated. We also found that amphetamine pretreatment altered mRNA expression for molecular markers associated with neuroinflammation and renin-angiotensin-aldosterone system (RAAS) activation in the lamina terminalis, a brain region implicated in the control of sympathetic nervous system tone and blood pressure. The results indicated amphetamine upregulated mRNA expression underlying neuroinflammation and, to a lesser degree, message for components of the RAAS in the lamina terminalis. However, we found no changes in mRNA expression in the paraventricular nucleus. These results suggest that a history of stimulant use may predispose individuals to developing hypertension by promoting neuroinflammation and upregulating activity of the RAAS in the lamina terminalis.

Keywords: amphetamine; angiotensin II; hypertension; lamina terminalis; neuroinflammation.

Publication types

  • Research Support, N.I.H., Extramural

MeSH terms

  • Amphetamine / pharmacology*
  • Angiotensin II / pharmacology
  • Animals
  • Blood Pressure / drug effects
  • Blood Pressure / physiology
  • Central Nervous System Stimulants / pharmacology*
  • Diet, High-Fat
  • Disease Models, Animal
  • Hypertension / chemically induced
  • Hypertension / physiopathology*
  • Hypothalamus / drug effects*
  • Hypothalamus / metabolism
  • Inflammation / drug therapy*
  • Paraventricular Hypothalamic Nucleus / drug effects
  • Rats

Substances

  • Central Nervous System Stimulants
  • Angiotensin II
  • Amphetamine