Bombesin stimulates inositol polyphosphate production in GH4C1 pituitary tumor cells: comparison with TRH

Biochem Biophys Res Commun. 1988 Jul 29;154(2):654-9. doi: 10.1016/0006-291x(88)90189-1.

Abstract

The hormones bombesin and thyrotropin-releasing hormone (TRH) stimulated formation of inositol- monophosphate, bisphosphate, trisphosphate and tetrakisphosphate with parallel time courses in GH4C1 cells, while a more polar inositol polyphosphate peak, consisting of inositol-pentakisphosphate and perhaps also inositol-hexakisphosphate, was unaffected by either hormone. Although bombesin and TRH had similar potencies in stimulating inositol trisphosphate production (Km = 30 nM and 40 nM, respectively), TRH was significantly more efficacious than bombesin. Maximal stimulation of inositol-1,4,5-trisphosphate formation by TRH was not further increased by addition of a maximally effective dose of bombesin, suggesting that the two hormones act through stimulation of a common pool of phospholipase C, and this enzyme pool can be fully stimulated by TRH, alone.

Publication types

  • Comparative Study
  • Research Support, Non-U.S. Gov't
  • Research Support, U.S. Gov't, P.H.S.

MeSH terms

  • Animals
  • Bombesin / pharmacology*
  • Cell Line
  • Inositol Phosphates / biosynthesis*
  • Kinetics
  • Pituitary Neoplasms / metabolism*
  • Rats
  • Sugar Phosphates / biosynthesis*
  • Thyrotropin-Releasing Hormone / pharmacology*

Substances

  • Inositol Phosphates
  • Sugar Phosphates
  • Thyrotropin-Releasing Hormone
  • Bombesin