Opioid use and dropout from extended-release naltrexone in a controlled trial: implications for mechanism

Addiction. 2020 Feb;115(2):239-246. doi: 10.1111/add.14735. Epub 2019 Aug 4.

Abstract

Background and aims: Extended-release formulations of naltrexone have emerged as effective treatment options for opioid use disorder. This post-hoc analysis examined the temporal relationship between episodes of opioid use and subsequent dropout in a placebo-controlled trial of extended-release injection naltrexone (XR-NTX) to draw inferences about the mechanism by which extended blockade of opioid receptors translates into clinical effectiveness.

Design: This was a 24-week multiple-site, double-blind, randomized trial of monthly XR-NTX versus placebo injections. We analyzed time to dropout from treatment using survival analysis with an extended Cox model as a function of treatment (XR-NTX versus placebo) and with weekly urine drug test (UDT) results for opioids at each week as a time-dependent covariate.

Setting: Thirteen addiction treatment programs in Russia, 2008-09.

Participants: A total of 250 adults with opioid use disorder who had completed in-patient detoxification.

Intervention: XR-NTX injection or placebo injection every 4 weeks with weekly clinic visits and biweekly counseling.

Measurements: Urine toxicology for opioids measured weekly and week of dropout from treatment.

Findings: The Cox model yielded a significant interaction of time-dependent urine toxicology by treatment (P = 0.024). Among patients receiving placebo, a positive UDT in a given week increased the risk for dropout from treatment in the subsequent week [hazard ratio (HR) = 6.25; 95% confidence interval (CI) = 3.6-10.0], whereas among patients receiving XR-NTX, a positive UDT result showed no significant effect on risk for dropout (HR = 1.67; 95% CI = 0.6-4.5). The proportion of patients who completed all 24 weeks without any positive UDT result was 31% on XR-NTX compared with 20% on placebo (P = 0.051).

Conclusions: Extended-release injection naltrexone was effective at reducing the risk of dropout from opioid use disorder treatment after an episode of opioid use. Just under a third of patients (31%) on XR-NTX had no opioid-positive urine tests across the trial, but the hypothesis that this would differ from placebo (20%) was not confirmed.

Keywords: Dropout; extended-release naltrexone; medication-assisted treatment; opioid dependence; opioid use disorder; relapse.

Publication types

  • Multicenter Study
  • Randomized Controlled Trial
  • Research Support, Non-U.S. Gov't

MeSH terms

  • Adult
  • Ambulatory Care
  • Delayed-Action Preparations / therapeutic use*
  • Double-Blind Method
  • Duration of Therapy
  • Female
  • Humans
  • Male
  • Naltrexone / therapeutic use*
  • Narcotic Antagonists / therapeutic use*
  • Opioid-Related Disorders / drug therapy*
  • Opioid-Related Disorders / urine
  • Patient Dropouts / statistics & numerical data*
  • Russia / epidemiology
  • Survival Analysis
  • Treatment Outcome

Substances

  • Delayed-Action Preparations
  • Narcotic Antagonists
  • Naltrexone