Copolymeric micelles as efficient inert nanocarrier for hypericin in the photodynamic inactivation of Candida species

Future Microbiol. 2019 Apr:14:519-531. doi: 10.2217/fmb-2018-0304. Epub 2019 Apr 29.

Abstract

Aim: To evaluate the efficacy of photodynamic inactivation (PDI) mediated by hypericin encapsulated in P-123 copolymeric micelles (P123-Hyp) alone and in combination with fluconazole (FLU) against planktonic cells and biofilm formation of Candida species Materials & methods: PDI was performed using P123-Hyp and an LED device with irradiance of 3.0 mW/cm2 . Results: Most of isolates (70%) were completely inhibited with concentrations up to 2.0 μmol/l of HYP and light fluence of 16.2 J/cm2. FLU-resistant strains had synergic effect with P123-HYP-PDI and FLU. The biofilm formation was inhibited in all species, in additional the changes in Candida morphology observed by scanning electron microscopy. Conclusion: P123-Hyp-PDI is a promising option to treat fungal infections and medical devices to prevent biofilm formation and fungal spread.

Keywords: spp.; biofilm; hypericin; photodynamic inactivation; resistance.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Anthracenes
  • Antifungal Agents / pharmacology*
  • Biofilms / drug effects*
  • Biofilms / growth & development
  • Biofilms / radiation effects
  • Candida / cytology
  • Candida / drug effects*
  • Candida / radiation effects
  • Drug Resistance, Fungal / drug effects
  • Drug Synergism
  • Drug Therapy, Combination
  • Fluconazole / pharmacology
  • Humans
  • Light
  • Micelles*
  • Microbial Sensitivity Tests
  • Microscopy, Electron, Scanning
  • Perylene / analogs & derivatives*
  • Perylene / pharmacology
  • Photochemotherapy / methods

Substances

  • Anthracenes
  • Antifungal Agents
  • Micelles
  • Perylene
  • hypericin
  • Fluconazole